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| (R*,R*)-N-[2-Hydroxy-5-[1-hydroxy-2-[[2-(4-methoxyphenyl)-1-methylethyl]amino]ethyl]phenyl]formamide fumarate dihydrate Basic information |
| (R*,R*)-N-[2-Hydroxy-5-[1-hydroxy-2-[[2-(4-methoxyphenyl)-1-methylethyl]amino]ethyl]phenyl]formamide fumarate dihydrate Chemical Properties |
Melting point | 116-120°C | storage temp. | 2-8°C | solubility | DMSO: soluble20mg/mL | form | solid | color | white to off-white | InChIKey | RATSWNOMCHFQGJ-XODSYJLDSA-N | CAS DataBase Reference | 183814-30-4 |
RIDADR | UN 2811 6.1 / PGII | WGK Germany | 3 | HS Code | 29242990 |
| (R*,R*)-N-[2-Hydroxy-5-[1-hydroxy-2-[[2-(4-methoxyphenyl)-1-methylethyl]amino]ethyl]phenyl]formamide fumarate dihydrate Usage And Synthesis |
Chemical Properties | Pale Yellow Solid | Uses | ForMoterol FuMarate Dihydrate is a selective β2-adrenergic receptor agonist,it is used as an antiasthmatic.
| Uses | A selective β2-adrenergic receptor agonist. Used as an antiasthmatic. | Uses | Formoterol is a selective β2-adrenergic receptor agonist. Formoterol is used as an antiasthmatic. | Biological Activity | Potent, selective and long-acting β 2 -adrenoceptor agonist. Displays 330-fold selectivity for β 2 over β 1 receptors (pK d values are 8.12 and 5.58 respectively). Potently relaxes guinea pig trachea (pD 2 = 9.29), and is longer-acting and 100-fold more potent than salbutamol. | Biochem/physiol Actions | β2-Adrenoreceptor agonist. |
| (R*,R*)-N-[2-Hydroxy-5-[1-hydroxy-2-[[2-(4-methoxyphenyl)-1-methylethyl]amino]ethyl]phenyl]formamide fumarate dihydrate Preparation Products And Raw materials |
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